Synthesis and Biological Characterization of Argyrin F

L Bülow, I Nickeleit, AK Girbig, T Brodmann, A Rentsch, U Eggert, F Sasse, H Steinmetz, R Frank, T Carlomagno, NP Malek & M Kalesse

ChemMedChem 5, 832–836 (2010)

Argyrin F unfolds its promising antitumor activity twice: First through stabilization of the tumor suppressor protein p27 and second by vascular damage.